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molstar

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A comprehensive macromolecular library.

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/** * Copyright (c) 2019-2020 mol* contributors, licensed under MIT, See LICENSE file for more info. * * @author Alexander Rose <alexander.rose@weirdbyte.de> * @author Fred Ludlow <Fred.Ludlow@astx.com> * * based in part on NGL (https://github.com/arose/ngl) */ import { __assign } from "tslib"; import { ParamDefinition as PD } from '../../../mol-util/param-definition'; import { AtomGeometryAngles, calcAngles, calcPlaneAngle } from '../chemistry/geometry'; import { Features } from './features'; import { typeSymbol, bondToElementCount, bondCount, formalCharge, compId, atomId } from '../chemistry/util'; import { ValenceModelProvider } from '../valence-model'; import { degToRad } from '../../../mol-math/misc'; import { ProteinBackboneAtoms } from '../../../mol-model/structure/model/types'; var GeometryParams = { distanceMax: PD.Numeric(3.5, { min: 1, max: 5, step: 0.1 }), backbone: PD.Boolean(true, { description: 'Include backbone-to-backbone hydrogen bonds' }), accAngleDevMax: PD.Numeric(45, { min: 0, max: 180, step: 1 }, { description: 'Max deviation from ideal acceptor angle' }), donAngleDevMax: PD.Numeric(45, { min: 0, max: 180, step: 1 }, { description: 'Max deviation from ideal donor angle' }), accOutOfPlaneAngleMax: PD.Numeric(90, { min: 0, max: 180, step: 1 }), donOutOfPlaneAngleMax: PD.Numeric(45, { min: 0, max: 180, step: 1 }), }; var HydrogenBondsParams = __assign(__assign({}, GeometryParams), { water: PD.Boolean(false, { description: 'Include water-to-water hydrogen bonds' }), sulfurDistanceMax: PD.Numeric(4.1, { min: 1, max: 5, step: 0.1 }) }); var WeakHydrogenBondsParams = __assign({}, GeometryParams); // // Geometric characteristics of hydrogen bonds involving sulfur atoms in proteins // https://doi.org/10.1002/prot.22327 // Satisfying Hydrogen Bonding Potential in Proteins (HBPLUS) // https://doi.org/10.1006/jmbi.1994.1334 // http://www.csb.yale.edu/userguides/datamanip/hbplus/hbplus_descrip.html function getUnitValenceModel(structure, unit) { var valenceModel = ValenceModelProvider.get(structure).value; if (!valenceModel) throw Error('expected valence model to be available'); var unitValenceModel = valenceModel.get(unit.id); if (!unitValenceModel) throw Error('expected valence model for unit to be available'); return unitValenceModel; } /** * Potential hydrogen donor */ function addUnitHydrogenDonors(structure, unit, builder) { var totalH = getUnitValenceModel(structure, unit).totalH; var elements = unit.elements; var _a = unit.model.atomicConformation, x = _a.x, y = _a.y, z = _a.z; var elementAromaticRingIndices = unit.rings.elementAromaticRingIndices; for (var i = 0, il = elements.length; i < il; ++i) { if (elementAromaticRingIndices.has(i)) continue; var element = typeSymbol(unit, i); if (( // include both nitrogen atoms in histidine due to // their often ambiguous protonation assignment isHistidineNitrogen(unit, i)) || (totalH[i] > 0 && (element === "N" /* N */ || element === "O" /* O */ || element === "S" /* S */))) { builder.add(4 /* HydrogenDonor */, 0 /* None */, x[elements[i]], y[elements[i]], z[elements[i]], i); } } } /** * Weak hydrogen donor. */ function addUnitWeakHydrogenDonors(structure, unit, builder) { var totalH = getUnitValenceModel(structure, unit).totalH; var elements = unit.elements; var _a = unit.model.atomicConformation, x = _a.x, y = _a.y, z = _a.z; for (var i = 0, il = elements.length; i < il; ++i) { if (typeSymbol(unit, i) === "C" /* C */ && totalH[i] > 0 && (bondToElementCount(structure, unit, i, "N" /* N */) > 0 || bondToElementCount(structure, unit, i, "O" /* O */) > 0 || inAromaticRingWithElectronNegativeElement(unit, i))) { builder.add(9 /* WeakHydrogenDonor */, 0 /* None */, x[elements[i]], y[elements[i]], z[elements[i]], i); } } } function inAromaticRingWithElectronNegativeElement(unit, index) { var _a = unit.rings, elementAromaticRingIndices = _a.elementAromaticRingIndices, all = _a.all; var ringIndices = elementAromaticRingIndices.get(index); if (ringIndices === undefined) return false; for (var i = 0, il = ringIndices.length; i < il; ++i) { var ring = all[ringIndices[i]]; for (var j = 0, jl = ring.length; j < jl; ++j) { var element = typeSymbol(unit, ring[j]); if (element === "N" /* N */ || element === "O" /* O */) { return true; } } } return false; } /** * Potential hydrogen acceptor */ function addUnitHydrogenAcceptors(structure, unit, builder) { var _a = getUnitValenceModel(structure, unit), charge = _a.charge, implicitH = _a.implicitH, idealGeometry = _a.idealGeometry; var elements = unit.elements; var _b = unit.model.atomicConformation, x = _b.x, y = _b.y, z = _b.z; var elementAromaticRingIndices = unit.rings.elementAromaticRingIndices; var add = function (i) { builder.add(5 /* HydrogenAcceptor */, 0 /* None */, x[elements[i]], y[elements[i]], z[elements[i]], i); }; for (var i = 0, il = elements.length; i < il; ++i) { if (elementAromaticRingIndices.has(i)) continue; var element = typeSymbol(unit, i); if (element === "O" /* O */) { // Basically assume all oxygen atoms are acceptors! add(i); } else if (element === "N" /* N */) { if (isHistidineNitrogen(unit, i)) { // include both nitrogen atoms in histidine due to // their often ambiguous protonation assignment add(i); } else if (charge[i] < 1) { // Neutral nitrogen might be an acceptor // It must have at least one lone pair not conjugated var totalBonds = bondCount(structure, unit, i) + implicitH[i]; var ig = idealGeometry[i]; if ((ig === 4 /* Tetrahedral */ && totalBonds < 4) || (ig === 3 /* Trigonal */ && totalBonds < 3) || (ig === 2 /* Linear */ && totalBonds < 2)) { add(i); } } } else if (element === "S" /* S */) { var resname = compId(unit, i); if (resname === 'CYS' || resname === 'MET' || formalCharge(unit, i) === -1) { add(i); } } } } function isWater(unit, index) { return unit.model.atomicHierarchy.derived.residue.moleculeType[unit.residueIndex[unit.elements[index]]] === 2 /* Water */; } function isBackbone(unit, index) { return ProteinBackboneAtoms.has(atomId(unit, index)); } function isRing(unit, index) { return unit.rings.elementRingIndices.has(index); } function isHistidineNitrogen(unit, index) { return compId(unit, index) === 'HIS' && typeSymbol(unit, index) === "N" /* N */ && isRing(unit, index); } function isBackboneHydrogenBond(unitA, indexA, unitB, indexB) { return isBackbone(unitA, indexA) && isBackbone(unitB, indexB); } function isWaterHydrogenBond(unitA, indexA, unitB, indexB) { return isWater(unitA, indexA) && isWater(unitB, indexB); } function isHydrogenBond(ti, tj) { return ((ti === 5 /* HydrogenAcceptor */ && tj === 4 /* HydrogenDonor */) || (ti === 4 /* HydrogenDonor */ && tj === 5 /* HydrogenAcceptor */)); } function isWeakHydrogenBond(ti, tj) { return ((ti === 9 /* WeakHydrogenDonor */ && tj === 5 /* HydrogenAcceptor */) || (ti === 5 /* HydrogenAcceptor */ && tj === 9 /* WeakHydrogenDonor */)); } function getGeometryOptions(props) { return { includeBackbone: props.backbone, maxAccAngleDev: degToRad(props.accAngleDevMax), maxDonAngleDev: degToRad(props.donAngleDevMax), maxAccOutOfPlaneAngle: degToRad(props.accOutOfPlaneAngleMax), maxDonOutOfPlaneAngle: degToRad(props.donOutOfPlaneAngleMax), }; } function getHydrogenBondsOptions(props) { return __assign(__assign({}, getGeometryOptions(props)), { includeWater: props.water, maxSulfurDistSq: props.sulfurDistanceMax * props.sulfurDistanceMax, maxDistSq: props.distanceMax * props.distanceMax }); } var deg120InRad = degToRad(120); function checkGeometry(structure, don, acc, opts) { var donIndex = don.members[don.offsets[don.feature]]; var accIndex = acc.members[acc.offsets[acc.feature]]; if (!opts.includeBackbone && isBackboneHydrogenBond(don.unit, donIndex, acc.unit, accIndex)) return; var donAngles = calcAngles(structure, don.unit, donIndex, acc.unit, accIndex); var idealDonAngle = AtomGeometryAngles.get(don.idealGeometry[donIndex]) || deg120InRad; if (donAngles.some(function (donAngle) { return Math.abs(idealDonAngle - donAngle) > opts.maxDonAngleDev; })) return; if (don.idealGeometry[donIndex] === 3 /* Trigonal */) { var outOfPlane = calcPlaneAngle(structure, don.unit, donIndex, acc.unit, accIndex); if (outOfPlane !== undefined && outOfPlane > opts.maxDonOutOfPlaneAngle) return; } var accAngles = calcAngles(structure, acc.unit, accIndex, don.unit, donIndex); var idealAccAngle = AtomGeometryAngles.get(acc.idealGeometry[accIndex]) || deg120InRad; // Do not limit large acceptor angles if (accAngles.some(function (accAngle) { return idealAccAngle - accAngle > opts.maxAccAngleDev; })) return; if (acc.idealGeometry[accIndex] === 3 /* Trigonal */) { var outOfPlane = calcPlaneAngle(structure, acc.unit, accIndex, don.unit, donIndex); if (outOfPlane !== undefined && outOfPlane > opts.maxAccOutOfPlaneAngle) return; } return true; } function testHydrogenBond(structure, infoA, infoB, distanceSq, opts) { var typeA = infoA.types[infoA.feature]; var typeB = infoB.types[infoB.feature]; if (!isHydrogenBond(typeA, typeB)) return; var _a = typeB === 5 /* HydrogenAcceptor */ ? [infoA, infoB] : [infoB, infoA], don = _a[0], acc = _a[1]; var donIndex = don.members[don.offsets[don.feature]]; var accIndex = acc.members[acc.offsets[acc.feature]]; // check if distance is ok depending on non-sulfur-containing hbond var maxDistSq = typeSymbol(don.unit, donIndex) === "S" /* S */ || typeSymbol(acc.unit, accIndex) === "S" /* S */ ? opts.maxSulfurDistSq : opts.maxDistSq; if (distanceSq > maxDistSq) return; if (!opts.includeWater && isWaterHydrogenBond(don.unit, donIndex, acc.unit, accIndex)) return; if (!checkGeometry(structure, don, acc, opts)) return; return 4 /* HydrogenBond */; } function testWeakHydrogenBond(structure, infoA, infoB, distanceSq, opts) { var typeA = infoA.types[infoA.feature]; var typeB = infoB.types[infoB.feature]; if (!isWeakHydrogenBond(typeA, typeB)) return; var _a = typeB === 5 /* HydrogenAcceptor */ ? [infoA, infoB] : [infoB, infoA], don = _a[0], acc = _a[1]; if (!checkGeometry(structure, don, acc, opts)) return; return 8 /* WeakHydrogenBond */; } // export var HydrogenDonorProvider = Features.Provider([4 /* HydrogenDonor */], addUnitHydrogenDonors); export var WeakHydrogenDonorProvider = Features.Provider([9 /* WeakHydrogenDonor */], addUnitWeakHydrogenDonors); export var HydrogenAcceptorProvider = Features.Provider([5 /* HydrogenAcceptor */], addUnitHydrogenAcceptors); export var HydrogenBondsProvider = { name: 'hydrogen-bonds', params: HydrogenBondsParams, createTester: function (props) { var maxDistance = Math.max(props.distanceMax, props.sulfurDistanceMax); var opts = getHydrogenBondsOptions(props); return { maxDistance: maxDistance, requiredFeatures: new Set([4 /* HydrogenDonor */, 5 /* HydrogenAcceptor */]), getType: function (structure, infoA, infoB, distanceSq) { return testHydrogenBond(structure, infoA, infoB, distanceSq, opts); } }; } }; export var WeakHydrogenBondsProvider = { name: 'weak-hydrogen-bonds', params: WeakHydrogenBondsParams, createTester: function (props) { var opts = getGeometryOptions(props); return { maxDistance: props.distanceMax, requiredFeatures: new Set([9 /* WeakHydrogenDonor */, 5 /* HydrogenAcceptor */]), getType: function (structure, infoA, infoB, distanceSq) { return testWeakHydrogenBond(structure, infoA, infoB, distanceSq, opts); } }; } }; //# sourceMappingURL=hydrogen-bonds.js.map